The Formestane Guide That You’ve Been Waiting For

Formestane is one of the prohormones that you’ll surely come across when you’re prepping up for your next cycle. But the question is will this compound really pull off the good stuff that it’s said to deliver? Let’s find out shortly in this through yet relaxed walkthrough.

So What is Formestane?

At its simplest, Formestane is a derivative of Androstenedione, which is more popularly known among bodybuilders and strength athletes as “andro.” Its only difference from andro is the addition of a 4-hydroxyl group in its chemical makeup. Besides being naturally produced in the body, particularly by the testes, adrenal glands as well as the ovaries, this compound is also present in meat and some plants.

Formestane chemical structure

Developed in the 1970’s by East German scientists to increase the power and endurance of their athletes during competitions, it is even said that Androstenedione was so potent that a single snort of this compound caused a massive spike in testosterone levels that lasted for as long as three (3) hours.  This is because andro almost immediately converts to testosterone as soon as it is metabolized by the body.

Alternatively, it is also said that Androstenedione was created to alleviate the effects and cure estrogen-receptor positive breast cancer in post-menopausal women, but made its way to the bodybuilding world along the way.

Metabolic pathway of Androstenedione

And given that snorting andro an hour before an event was a team requirement by the East Germans in the 1988 Olympics, it isn’t that tricky to figure out why they gathered quite an impressive haul during the same.

This prohormone has gathered a loyal following in the bodybuilding world over the years for its convenient modes of administration as well as the rapid results that it can trigger when cycled –not mentioning the free endorsement courtesy of MLB All-Star Mark “Big Mac” McGwire when he was still playing as first baseman for the St. Louis Cardinals.

Considered by seasoned prohormone users as a potent performance enhancer and recovery booster, Formestane is usually available in four forms, namely gel, powder, capsule and spray, which offer a whole lot of difference in terms of convenience compared to injectables. Interestingly, an injectable version of Formestane called Lentaron was also produced one time, but has been since withdrawn in the market.

Experts emphasize that the beneficial effects of the spray can kick in at approximately half an hour, and the powder and capsule at around two hours. The gel form can take a bit longer to get in action compared to its counterparts, but still quite strong in terms of efficacy.

Aside from its prohormone capabilities, Formestane is also a known selective irreversible steroidal aromatase inhibitor with the chemical designation 4- Hydroxyandrost-4-ene-3,17-dione.

It basically blocks estrogen conversion in the body, which is definitely a plus if you’re steering clear from nasty estrogenic issues like gynecomastia and tenderness in and around the breast area during or after a cycle. However, it is still recommended that you have a proper post cycle therapy or PCT to keep these issues at bay.

What Positive Effects Does Formestane Have?

According to seasoned prohormone users, cycling with Formestane stimulates faster fat loss and a considerable boost in strength levels and muscle mass.

Using this compound also causes an increase in the amount of red blood cells in the body, which results to a faster delivery of oxygen in the bloodstream. This means you will last way longer than usual during a workout. You’ll also keep clear from the catabolic effects of heavy training while at it.

Some bodybuilders and strength athletes who have already given Formestane a go also report that their mood and aggression considerably improved when they cycled with this prohormone.

Does Formestane Have Side Effects?

Now while the risk of being vulnerable to side effects when cycling with prohormones is significantly lower compared to using straight up anabolic steroids, there are still a few potential issues that could get in the picture if you’re not keeping a close eye on your dosage and cycling time or perhaps not having the right on-cycle support.

According to experts, these issues include the following:

  • Unexpected mood swings
  • Hirsutism and masculinization in women
  • Testicular atrophy
  • Sudden onset of acne

The Recommended Dosage and Cycling of Formestane

According to veteran prohormone users, the ideal dosage of Formestane when you’re using it for aromatase inhibition is 150 milligrams to 250 milligrams every day via oral administration and 100 milligrams to 200 milligrams if it’s used through transdermal means.

Moreover, topical gel application should be between 100 milligrams to 200 milligrams. The gel should be applied vigorously on the upper arms and thighs thoroughly and must be allowed to dry completely around 5 minutes before doing other activities.

When you’re looking to use Formestane for anabolic effects, a daily dose of 800 milligrams to 1,000 milligrams should be taken. A typical cycle length of Formestane is between 2 to 4 weeks. This compound has a half-life of 4 days.

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