The Complete Guide on Superdrol

There is a very big possibility that Superdrol is on your list of prohormones to consider when it comes to serious size, strength and mass gains.

But the thing is if you’re still a bit unsure that this one is really the choice you’d have to go for, make sure you follow along to find out more about this very successful prohormone that took the bodybuilding world by storm in the last decade.

What is Superdrol?

Let’s start things off by clarifying one rather popular misconception. Superdrol is not the name of the compound that makes this prohormone tick, but is actually the brand name it was marketed under when it was released by Designer Supplements LLC in 2005. There are also accounts that Anabolic Extreme originally dubbed the name for a nutritional supplement it launched during the same time.

A sample of Superdrol released by Designer Supplements LLC
A sample of Superdrol released by Designer Supplements LLC

Interestingly, the name “Superdrol” is a play on words to give bodybuilders the notion that it’s the stuff they should zero in on if they’re gunning for fast and solid results. It’s supposed to be a combination of “Super” and “Anadrol,” which was then considered as the most powerful mass builder on the market.

The active compound in Superdrol is methasterone (systematic IUPAC name: 17β-Hydroxy-2α,17α-dimethyl-5α-androstane-3-one) – also known as methyldrostanolone and methasteron – which rose to superstar status during its run for the speedy results it can deliver when cycled, especially in terms of very hard and dry gains just after a couple of weeks of usage. Reports of achieving upwards of 20 to 30 pounds of muscle mass were not uncommon from users after cycling with Superdrol in the span of 4 weeks. Its half-life is timed at 6 to 8 hours.

The chemical structure of Superdrol
The chemical structure of Superdrol

Besides the considerable boost in size and mass, this dihydrotestosterone or DHT-derived prohormone has also been seen to have the ability to take strength levels up a notch. Based on user logs, they were able to increase their overall lifts by as much as 20 to 25 percent in just the second week of their cycle with this compound.

At its simplest, Superdrol’s power and intensity comes from its being similar with Masteron, a different type of anabolic steroid, but without the ester chain that the latter flaunts in its chemical structure. It works by optimizing the body’s ability to retain nitrogen and its synthesis of protein, which result to not just gains in size, mass, strength and endurance, but also the speed muscles recover after going through a grueling workout.

Plus, its androgenic activity in the body was much lower compared to its prohormone counterparts. This means that Superdrol doesn’t put you at risk of experiencing increased hair loss or hair growth as well as bouts of acne when you use it compared to other anabolic steroids. It isn’t necessary to use an anti-estrogen when cycling with this compound as well.

Superdrol before and after
Superdrol before and after

During its short run when Superdrol was still freely available on the shelves, this orally ingested prohormone was considered as a crucial bulking, cutting and recovery agent that yielded quick results without having to do anything with needles. This was the biggest reason why it’s earned a lot of loyal followers worldwide.

On the other hand, Superdrol is basically a type of C17-aa anabolic steroid and can be toxic to the liver, especially when used without the proper on-cycle support and post cycle therapy. Clinical researchers emphasize that cycling with this prohormone can trigger the values of liver enzymes to surge, which indicates stress and can lead to health issues if not given the right attention it deserves.

Now while Superdrol has become quite a legend in the prohormone world, it was banned by the U.S. Food and Drug Administration (FDA) in 2006, which forced its manufacture and distribution to halt. However, the ban did not stop the production and sale of the methasterone compound in both legal consumer over-the-counter market and underground channels.

The FDA cracked down on this further by classifying the prohormone as a Schedule III controlled substance, along with other anabolic steroids, in August 29, 2012. There are still Superdrol “clones” that you can get your hands on these days, though. And they’ve been on the black market ever since.

After this prohormone’s ban took effect in 2012, many of its users picked Dymethazine as an alternative. Dymethazine is made up of two Superdrol molecules that are kept together by a single nitrogen atom. It was spared from the ban because it had an entirely different hormonal structure.

The chemical structure of Dymethazine
The chemical structure of Dymethazine


Although Superdrol was launched in the market as a “designer steroid” in 2005, its active compound, methasterone, has already been formulated in 1956 by the Syntex Corporation as a component to develop a compound that has the ability to stave off tumors.

Besides pointing out its anti-tumor properties, methasterone was also described in a scientific article in 1959 as being a “potent orally active anabolic agent” with a weak androgenic activity. Subsequent articles on the compound emphasized that it shared an oral bioavailability akin to methyl-testosterone and scored a very high anabolic to androgenic ratio or “Q-ratio” of 20.

However, methasterone did not fully become a prescription drug even with its proven attributes. The Syntex Corporation instead focused on developing a non-17α-alkylated counterpart of this compound called drostanolone and eventually released it in the market as Masteron. It wasn’t until 2005 that methasterone – in the form of Superdrol – hit the shelves as a dietary supplement, which didn’t take long for it to become a huge success.


If you’re planning to integrate Superdrol in your bodybuilding checklist, here are the benefits that you will be in for:

  • Helps boost size and mass gains
  • Increases overall strength levels
  • Boosts nitrogen retention and protein synthesis
  • Can be used without an anti-estrogen
  • Doesn’t have as much androgenic activity compared to its counterparts
  • Can yield up to 30 pounds of lean muscle in 4 weeks
  • Acts really fast

Side Effects

Although Superdrol has been seen to have lower androgenic levels compared to other prohormones in the market, you can still be vulnerable to the following when you cycle with it:

  • Can cause a spike in blood pressure and bad cholesterol levels
  • Can place the body in a low testosterone state
  • Can be toxic to the liver without the proper support and precautions

A Quick Rundown on a Superdrol Cycle

Perhaps the most important guideline that you should keep in mind to make your cycle with Superdrol as successful as possible is having an idea of the right dosage to get you on track to achieving your goals. Here is a quick guide that you can use to kick off your cycle with this prohormone:

Dosage and Post Cycle Therapy (PCT) Pointers

It is very important to take note that Superdrol should be dosed low during the start of a cycle. Experienced users highly recommend that you begin with a daily dose of 10mg for the first week and increase your dosage to 20mg in the second and third weeks. It’s crucial that you take Superdrol daily with food. If you are very tolerant to this compound, you can bump up to 40mg in the fourth week.

A proper post cycle therapy should be carried out in the succeeding fifth to eighth weeks.

Moreover, experienced Superdrol users suggest that this compound stacks quite well with most anabolic steroids. Stacking some form of testosterone with this prohormone considerably improves realizing your cutting and bulking goals. Trenbolone is highly recommended with Superdrol when cutting, while Nandrolone is a nice choice to go with this compound during a bulking phase.

6 thoughts on “The Complete Guide on Superdrol

  1. Pingback: The Best Prohormones of 2016 and into 2017

  2. Alex Dupree says:

    Wanting to know if you bank transfers, as W. U is starting to get nosey waiting to know to much info. to transfer cash, money gram does dome times to depending on who it it on the phone, i just logged on your site but I hav’nt signed up yet, do I just use email and password, thz Flex

  3. Alex Duptee says:

    I sent email thing to sign up with to get superdrol, give the sign up details if you sell this product thz I wasn’t able sign on your date for dome reason, th, Alex

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